平安! 发表于 2011-11-9 19:57
4 |9 E- w2 Z9 L5 c+ i2 W: D: K9 WPazopanib (100 mg/kg/day free base equivalent) ) U9 A/ x. [( ^: C1 [
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。: m' w1 A# V5 U6 j! ]
搜索了一下,原料一大堆。$ n5 U5 O2 g7 l4 d6 {$ H; Q% S
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对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。" u% C1 e/ Y- r; O$ q0 `
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--------------------- DOSAGE AND ADMINISTRATION ----------------
! ]3 Z) R, k+ Z2 g% Z% ^* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
$ x) U7 J9 O; p3 ~0 e6 }* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
1 a5 p- W7 ^( V---------------------DOSAGE FORMS AND STRENGTHS --------------1 |/ h1 o. b! z. }& P6 U* s
200 mg tablets. (3)
5 [* \. ^) k3 P* Y' N. {-------------------------------CONTRAINDICATIONS------------------------ |