平安! 发表于 2011-11-9 19:57
3 G% \6 m6 _% Q' hPazopanib (100 mg/kg/day free base equivalent) 9 |2 K! n B% Z; u. f- {' q/ i* d, M
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。, ]( q8 E' Q! Z- E* D. `# ^
搜索了一下,原料一大堆。% F" X/ j+ \: \' K
( j1 y2 J, R; _+ z2 ]5 G& d6 t8 _对不起!100mg/kg是用于移植瘤的,我弄错了。1 U; L) E! G8 ?" K
4 V) i( s( V6 z) Q' U以下是正版说明书的推荐用量。' {' z1 G3 h1 W, `/ X8 |- k1 `
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--------------------- DOSAGE AND ADMINISTRATION ----------------, `9 L4 f6 G- C: B* H1 {
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) . d2 i ~% F4 k
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) ( D7 r: r7 x9 U
---------------------DOSAGE FORMS AND STRENGTHS --------------
0 p8 o! W0 Y( V- A3 ^; Q- V/ x200 mg tablets. (3)
/ F/ L4 [# U9 ~: z-------------------------------CONTRAINDICATIONS------------------------ |